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Cayman Gk241; 5 Mg; 1899930-93-8; ≥98%
List Price
$249.00
Your Price
$249.00
Cayman Gk241; 5 Mg; 1899930-93-8; ≥98% - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-37689-5
MFG.PART:
37689-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
GK241 is a secretory phospholipase A2 (sPLA2) (Type IIA) inhibitor (IC50s = 0.143 and 0.068 µM for the human and mouse enzymes, respectively).1,2 It inhibits IL-1β-induced production of prostaglandin E2 (PGE2; Item No. 14010) in isolated rat renal mesangial cells when used at concentrations of 3 and 10 µM.3 GK241 also inhibits the severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) main protease (Mpro), also known as 3C-like protease (3CLpro; IC50 = 24 µM).1
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-(1,2-dioxo
CAS Number
1899930-93-8
Molecular Formula
C21H39NO4
Formula Weight
369.5
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: Slightly soluble
- DMSO: 2 mg/ml
- Ethanol: 1 mg/ml
λmax
244 nm
SMILES
CCCCCCCCCCCCCCC(C(N[C@H](C(O)=O)C(C)C)=O)=O
InChi Code
InChI=1S/C21H39NO4/c1-4-5-6-7-8-9-10-11-12-13-14-15-16-18(23)20(24)22-19(17(2)3)21(25)26/h17,19H,4-16H2,1-3H3,(H,22,24)(H,25,26)/t19-/m0/s1
InChi Key
ZVJNWONHYXBMJL-IBGZPJMESA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 2 years
| SKU | CAYM-37689-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 37689-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1899930-93-8 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |