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Cayman L-Glutamine-D5, 5mg
List Price
$249.00
Your Price
$249.00
Cayman L-Glutamine-D5, 5mg - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-34839-5
MFG.PART:
34839-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
CID-16020046 is a GPR55 inverse agonist that antagonizes GPR55 constitutive activity with an IC50 value of 15 μM. It inhibits GPR55-mediated ERK1/2 phosphorylation, LPI-induced Ca2+ signaling (IC50 = 0.21 μM in HEK-GPR55 cells), and GPR55-mediated transcription factor activation. It does not affect ERK1/2 phosphorylation or transcription factor activation in CB receptor expressing cells and demonstrates weak activity against a broad spectrum of other GPCRs, ion channels, kinases, and nuclear receptors. This compound has been shown to block GPR55-mediated endothelial wound healing and reverse LPI-inhibited platelet aggregation.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
4-[4,6-dihydro-
CAS Number
834903-43-4
Molecular Formula
C25H19N3O4
Formula Weight
425.4
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 25 mg/ml
- DMSO: 25 mg/ml
λmax
280 nm
SMILES
OC(C(C=C1)=CC=C1N2C(C3=CC=CC(O)=C3)C4=C(NN=C4C5=CC=C(C)C=C5)C2=O)=O
InChi Code
InChI=1S/C25H19N3O4/c1-14-5-7-15(8-6-14)21-20-22(27-26-21)24(30)28(18-11-9-16(10-12-18)25(31)32)23(20)17-3-2-4-19(29)13-17/h2-13,23,29H,1H3,(H,26,27)(H,31,32)
InChi Key
VGUQVYZXABOXCX-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-34839-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 34839-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | Canada |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 14341-78-7 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |