Cayman Azd 8931; Purity- Greater Than Or Equal To 98%; Size- 10 M

Name: Cayman Azd 8931; Purity- Greater Than Or Equal To 98%; Size- 10 M
SKU: CAYM-24196-10
Price: 235.00 USD

List Price $235.00 Your Price $235.00

Cayman Azd 8931; Purity- Greater Than Or Equal To 98%; Size- 10 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)

NETA PART: CAYM-24196-10

MFG.PART: 24196-10

UNSPSC: 12352200

Manufacturer: Cayman

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Description

Product Description

Azamulin is a selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC₅₀ values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources). It is at least 50-fold less potent against CYP2J2 and 100-fold less effective against all other CYP isoforms. Azamulin potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.^,

WARNING This product is not for human or veterinary use.

Technical Information

Formal Name

(3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester 2-[(3-amino-1H-1,2,4-triazol-5-yl)thio]-acetic acid

CAS Number

76530-44-4

Synonyms

Antibiotic TDM 85-530
SA 85530b

Molecular Formula

C₂₄H₃₈N₄O₄S

Formula Weight

478.7

Purity

≥98%

Formulation

A crystalline solid

Solubility

DMF: 30 mg/ml
DMSO: 30 mg/ml
Ethanol: 30 mg/ml
Ethanol:PBS(pH 7.2) (1:1): 0.5 mg/ml

SMILES

O=C1CC[C@@]23[C@@H](C)[C@H](O)[C@@](CC)(C)C[C@@H](OC(CSC4=NN=C(N)N4)=O)[C@](C)([C@H](C)CC3)[C@@]21[H]

InChi Code

InChI=1S/C24H38N4O4S/c1-6-22(4)11-16(32-17(30)12-33-21-26-20(25)27-28-21)23(5)13(2)7-9-24(14(3)19(22)31)10-8-15(29)18(23)24/h13-14,16,18-19,31H,6-12H2,1-5H3,(H3,25,26,27,28)/t13-,14+,16-,18+,19+,22-,23+,24+/m1/s1

InChi Key

FMHQJXGMLMSMLC-WBUYAQKGSA-N

Shipping & Storage Information

Storage

-20°C

Shipping

Room Temperature in continental US; may vary elsewhere

Stability

≥ 4 years

Specifications

More Information
SKU	CAYM-24196-10
Featured	No
Supplier Part Number	24196-10
UM	EA
UNSPSC	12352200
Manufacturer Name	Cayman
MSDS URL	Click here
Temperature	-20
Refrigerated-Frozen	Refrigerated
CountryOfOrigin	China
ProductLine	CAYM
Qty	1
MinOrderQty	1
Weight	7.000000
Lead Time	2
Hazardous	N
CAS Number	848942-61-0
Energy Star	No
Green	No
ACT Ecolabel	No
Controlled	N

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NETA PART NO.	Quantity

Cayman Azd 8931; Purity- Greater Than Or Equal To 98%; Size- 10 M

Product Description

Technical Information

Shipping & Storage Information

Product Title