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Cayman Mle-4901; Purity- Greater Than Or Equal To 98%; Size- 5 Mg
List Price
$268.00
Your Price
$268.00
Cayman Mle-4901; Purity- Greater Than Or Equal To 98%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-23587-5
MFG.PART:
23587-5
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
MLE-4901 is an antagonist of the neurokinin-3 (NK3) receptor.1 It inhibits human liver microsomal CYP3A4/5 with apparent IC50 values of 7.1 and 19.8 μM in midazolam 1-hydroxylation and testosterone 6β-hydroxylation assays, respectively.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
3-[(methyl sulfonyl)amino]- 2-phenyl-N- [(1S)-1-phenyl propyl]-4- quinoline carboxamide
CAS Number
941690-55-7
Synonyms
- AZD 2624
- AZD 4901
Molecular Formula
C26H25N3O3S
Formula Weight
459.6
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
- DMF: 30mg/mL
- DMF:PBS (pH 7.2) (1:3): 0.25mg/mL
- DMSO: 20mg/mL
λmax
236 nm
SMILES
CS(NC1=C(C(N[C@H](C2=CC=CC=C2)CC)=O)C3=CC=CC=C3N=C1C4=CC=CC=C4)(=O)=O
InChi Code
InChI=1S/C26H25N3O3S/c1-3-21(18-12-6-4-7-13-18)28-26(30)23-20-16-10-11-17-22(20)27-24(19-14-8-5-9-15-19)25(23)29-33(2,31)32/h4-17,21,29H,3H2,1-2H3,(H,28,30)/t21-/m0/s1
InChi Key
QYTBBBAHNIWFOD-NRFANRHFSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-23587-5 |
|---|---|
| Featured | No |
| Supplier Part Number | 23587-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | United States |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 941690-55-7 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |