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Cayman Formoterol-13c-D3 (Hemifumarate); Purity- Greater Than Or
List Price
$183.00
Your Price
$183.00
Cayman Formoterol-13c-D3 (Hemifumarate); Purity- Greater Than Or Equal To 99% Deuterated Forms (D1-D3); Size- 500 Micrograms; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-25317-500
MFG.PART:
25317-500
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
Formoterol-13C-d3 is intended for use as an internal standard for the quantification of formoterol (Item No. 15584) by GC- or LC-MS. Formoterol is a selective agonist of the β2-adrenergic receptor (β2-AR; Kis = 7.58 and 2,630 nM for β2- and β1-ARs, respectively).1 It is selective for β-ARs in isolated guinea pig trachea over those in atrial tissue (pD2s = 9.29 and 6.98, respectively) and has a long duration of action.2,1 Aerosolized formoterol (10 µg/ml, inhaled) prevents the late asthmatic response and eosinophil and macrophage infiltration in bronchoalveolar lavage fluid (BALF), and as well as reduces bronchial reactivity in a guinea pig model of allergic asthma induced by ovalbumin.3 Formulations containing formoterol have been used, alone and in combination with other compounds, in the treatment of chronic obstructive pulmonary disease and asthma.4,5,6
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
rel-N-[2-hydroxy-
Molecular Formula
C18[13C]H21D3N2O4 • 1/2C4H4O4
Formula Weight
406.5
Purity
≥99% deuterated forms (d1-d3)
Formulation(Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
- DMSO: 20 mg/ml
- Methanol: 1 mg/ml
- Water: Slightly Soluble
SMILES
OC(C=C1)=C(NC([H])=O)C=C1[C@H](O)CN[C@@H](C)CC2=CC=C(O[13C]([2H])([2H])[2H])C=C2.OC(/C=C/C(O)=O)=O
InChi Code
InChI=1S/2C19H24N2O4.C4H4O4/c2*1-13(9-14-3-6-16(25-2)7-4-14)20-11-19(24)15-5-8-18(23)17(10-15)21-12-22;5-3(6)1-2-4(7)8/h2*3-8,10,12-13,19-20,23-24H,9,11H2,1-2H3,(H,21,22);1-2H,(H,5,6)(H,7,8)/b;;2-1+/t2*13-,19+;/m00./s1/i2*2+1D3;
InChi Key
OBRNDARFFFHCGE-RPXDEYMZSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-25317-500 |
|---|---|
| Featured | No |
| Supplier Part Number | 25317-500 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | Canada |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |