We use cookies to make your experience better. To comply with the new e-Privacy directive, we need to ask for your consent to set the cookies. Learn more.
Cayman Itraconazole-D5; Purity- Greater Than Or Equal To 99% Deut
List Price
$330.00
Your Price
$330.00
Cayman Itraconazole-D5; Purity- Greater Than Or Equal To 99% Deuterated Forms (D1-D5); Size- 1 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
NETA PART:
CAYM-25219-1
MFG.PART:
25219-1
UNSPSC:
12352200
Manufacturer:
Cayman
Product Description
CH5138303 is a triazine Hsp90 inhibitor. CH5138303 binds to the N-terminus of Hsp90α (Kd = 0.52 nM) and inhibits growth of HCT116 and NCI-N87 human tumor cell lines in vitro (IC50s = 89 and 66 nM, respectively). CH5138303 also inhibits growth of human NCI-N87 gastric cancer xenografts (ED50 = 3.9 mg/kg) and displays high oral bioavailability in mice.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
4-[[4-amino- 6-(5-chloro- 1H,3H-naphtho [1,8-cd]pyran- 6-yl)-1,3,5- triazin-2-yl] thio]-butanamide
CAS Number
959763-06-5
Molecular Formula
C19H18ClN5O2S
Formula Weight
415.9
Purity
≥99%
Formulation
A crystalline solid
Solubility
- DMF: 33 mg/ml
- DMSO: 33 mg/ml
- DMSO:PBS (pH 7.2)(1:5): 0.16 mg/ml
λmax
229 nm
SMILES
NC1=NC(SCCCC(N)=O)=NC(C2=C(Cl)C=C3C4=C2C=CC=C4COC3)=N1
InChi Code
InChI=1S/C19H18ClN5O2S/c20-13-7-11-9-27-8-10-3-1-4-12(15(10)11)16(13)17-23-18(22)25-19(24-17)28-6-2-5-14(21)26/h1,3-4,7H,2,5-6,8-9H2,(H2,21,26)(H2,22,23,24,25)
InChi Key
VIGHQZSTZWNWFA-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-25219-1 |
|---|---|
| Featured | No |
| Supplier Part Number | 25219-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer Name | Cayman |
| MSDS URL | Click here |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | Canada |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.000000 |
| Lead Time | 2 |
| Hazardous | N |
| CAS Number | 1217510-38-7 |
| Energy Star | No |
| Green | No |
| ACT Ecolabel | No |
| Controlled | N |