Cayman Stictic Acid; Purity- Greater Than Or Equal To 95%; Size-

Arachidonoyl-2-fluoroethylamide (2-fluoro AEA) is an analog of anandamide in which the alcohol of the ethanolamide group has been removed and replaced with a fluorine atom. This substitution adds considerably increased binding affinity for the CB₁ receptor (K_is = 26.7 and 908 nM for CB₁ and CB₂, respectively). It also contributes additional selectivity, in that binding to CB₂ is decreased relative to AEA. However, the in vivo activity of 2-fluoro AEA is enhanced much less than the binding affinity, because the analog remains a good substrate for FAAH and is rapidly hydrolyzed by this enzyme.

WARNING This product is not for human or veterinary use.